Open access
Aug 2026
Identification, Structure–Activity Relationship (SAR), and Biological Evaluation of New Chemical Series as Malaria Parasite PfGCN5 Bromodomain Inhibitors
Despite considerable progress in prevention, treatment, and eradication efforts, malaria continues to impose a significant public health and socioeconomic burden for many countries around the globe. With the effectiveness of current treatment options partially or totally compromised due to resistance, the validation of...
Pedro Martín-Acosta, Abbas H. K. Al Temimi, Luma Godoy Magalhaes et al.
· ACS Omega · 0 citations