Open access
Aug 2026
Building TIPE2 Inhibitors from Quadrant System for Fragment-Based Docking
It is demonstrated that quadrant-based fragment docking provides an effective strategy for designing inhibitors targeting proteins with large binding cavities and provides promising lead compounds for the development of TIPE2 inhibitors.
Dorothea West, Pearl Miller, Jerica Wilson et al.
· The Scientist · 0 citations