Aug 2026
Striking two targets with one scaffold via benzo[d]imidazole-isatin conjugates as potent dual VEGFR-2/c-MET antagonists.
Chemical 8b may serve as a promising candidate for further anticancer research after demonstrating encouraging dual kinase inhibitory action and exhibiting a favorable selectivity profile for normal MCF-10A cells.
Mohamed El-Naggar, Rofaida Salem, Mona M. Kabeel et al.
· Bioorganic & Medicinal Chemi... · 0 citations